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    Kinesin spindle protein (KSP) inhibitors. 9. Discovery of (2S)-4-(2,5-difluorophenyl)-n-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide (MK-0731) for the treatment of taxane-refractory cancer (English)
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    Christopher D Cox
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    Paul J Coleman
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    Michael J Breslin
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    David B Whitman
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    Robert M Garbaccio
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    Mark E Fraley
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    Carolyn A Buser
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    Eileen S Walsh
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    Kelly Hamilton
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    Michael D Schaber
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    Robert B Lobell
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    Weikang Tao
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    Joseph P Davide
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    Ronald E Diehl
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    Marc T Abrams
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    Vicki J South
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    Hans E Huber
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    Maricel Torrent
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    Thomayant Prueksaritanont
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    Chunze Li
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    Donald E Slaughter
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    Elizabeth Mahan
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    Carmen Fernandez-Metzler
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    Youwei Yan
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    Lawrence C Kuo
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    Nancy E Kohl
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    George D Hartman
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    24 July 2008
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    51
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    4239-52
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    14
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