Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator (Q27622313)

2

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C Luong

3

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K Radika

4

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A Martelli

5

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P A Sprengeler

6

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J Wang

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H Chan

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L Wong

On the size of the active site in proteases. I. Papain

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publication date

April 2000

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published in

Chemistry and Biology

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volume

7

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issue

4

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page(s)

299-312

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cites work

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Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: implications for the inhibition of factor Xa, tPA, and urokinase.

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Rational design and synthesis of novel, potent bis-phenylamidine carboxylate factor Xa inhibitors

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Design of benzamidine-type inhibitors of factor Xa

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X-ray structure of active site-inhibited clotting factor Xa. Implications for drug design and substrate recognition

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The urokinase-type plasminogen activator system in cancer metastasis: a review

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The 2.3 A crystal structure of the catalytic domain of recombinant two-chain human tissue-type plasminogen activator

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7 January 2021

The crystal structure of the catalytic domain of human urokinase-type plasminogen activator

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Recruiting Zn2+ to mediate potent, specific inhibition of serine proteases

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The Protein Data Bank: a computer-based archival file for macromolecular structures

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Purification of urokinase by affinity chromatography

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Program DYNAFIT for the analysis of enzyme kinetic data: application to HIV proteinase

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6 Statistical analysis of enzyme kinetic data

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Structure of the hirugen and hirulog 1 complexes of alpha-thrombin

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Crystal structure of recombinant human tissue kallikrein at 2.0 A resolution

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Structure of human des(1-45) factor Xa at 2.2 A resolution

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The isomorphous structures of prethrombin2, hirugen-, and PPACK-thrombin: changes accompanying activation and exosite binding to thrombin

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Episelection: novel Ki approximately nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface

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7 January 2021

10.1016/S1074-5521(00)00104-6

Identifiers

DOI

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Fatcat ID

release_523fr7de7ncpxmcyu6ghertjca

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/523fr7de7ncpxmcyu6ghertjca

24 November 2022