Quantitative structure-agonist activity relationship of capsaicin analogues (Q71749035)

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20 October 2019

title

Quantitative structure-agonist activity relationship of capsaicin analogues (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:7561979%20AND%20SRC:MED&resulttype=core&format=json

20 October 2019

author name string

G Klopman

series ordinal

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:7561979%20AND%20SRC:MED&resulttype=core&format=json

20 October 2019

J Y Li

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:7561979%20AND%20SRC:MED&resulttype=core&format=json

20 October 2019

publication date

1 June 1995

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:7561979%20AND%20SRC:MED&resulttype=core&format=json

Journal of Computer - Aided Molecular Design

20 October 2019

language of work or name

English

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published in

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:7561979%20AND%20SRC:MED&resulttype=core&format=json

20 October 2019

volume

9

1 reference

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20 October 2019

issue

3

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20 October 2019

page(s)

283-294

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Cellular mechanism of action of resiniferatoxin: a potent sensory neuron excitotoxin

20 October 2019

cites work

1 reference

12 December 2020

Mechanisms and therapeutic potential of vanilloids (capsaicin-like molecules).

1 reference

12 December 2020

Competitive inhibition by capsazepine of [3H]resiniferatoxin binding to central (spinal cord and dorsal root ganglia) and peripheral (urinary bladder and airways) vanilloid (capsaicin) receptors in the rat

1 reference

12 December 2020

Analogues of capsaicin with agonist activity as novel analgesic agents; structure-activity studies. 1. The aromatic "A-region".

1 reference

12 December 2020

Sensory neuron-specific actions of capsaicin: mechanisms and applications

1 reference

12 December 2020

Sensory effects of capsaicin congeners I. Relationship between chemical structure and pain-producing potency of pungent agents

1 reference

12 December 2020

Application of liquid chromatography with on-line radiochemical detection to metabolism studies on a novel class of analgesics

1 reference

12 December 2020

META. 1. A program for the evaluation of metabolic transformation of chemicals

1 reference

12 December 2020

Pharmacologic actions of capsaicin: Apparent involvement of substance P and serotonin

1 reference

12 December 2020

Analogues of capsaicin with agonist activity as novel analgesic agents; structure-activity studies. 2. The amide bond "B-region"

1 reference

12 December 2020

Inhibition of [3H]resiniferatoxin binding to rat dorsal root ganglion membranes as a novel approach in evaluating compounds with capsaicin-like activity

1 reference

12 December 2020

Temperature-dependence of the action of nerve blocking agents and its relationship to membrane-buffer partition coefficients: thermodynamic implications for the site of action of local anaesthetics

1 reference

12 December 2020

Vanilloids. 1. Analogs of capsaicin with antinociceptive and antiinflammatory activity

1 reference

12 December 2020

Hydrophobicity and central nervous system agents: on the principle of minimal hydrophobicity in drug design

1 reference

12 December 2020

Analogues of capsaicin with agonist activity as novel analgesic agents; structure-activity studies. 3. The hydrophobic side-chain "C-region".

1 reference

12 December 2020

Long-lasting agonist activity produced by a capsaicin-like photoaffinity probe

1 reference

12 December 2020

Molecular target size of the vanilloid (capsaicin) receptor in pig dorsal root ganglia

1 reference

12 December 2020

The vanilloid (capsaicin) receptor: receptor types and species differences

1 reference

12 December 2020

Capsaicin-induced ion fluxes in dorsal root ganglion cells in culture

1 reference

12 December 2020

Cardiovascular interactions of nonivamide, glyceryl nonivamide, capsaicin analogues, and substance P antagonist in rats.

1 reference

12 December 2020

Estimation of aqueous solubility of organic molecules by the group contribution approach. Application to the study of biodegradation

1 reference

12 December 2020

Molecular mechanisms of local anesthesia: a review

1 reference

12 December 2020

The discovery of capsazepine, the first competitive antagonist of the sensory neuron excitants capsaicin and resiniferatoxin

1 reference

12 December 2020

Resiniferatoxin and its analogs provide novel insights into the pharmacology of the vanilloid (capsaicin) receptor

1 reference

12 December 2020

Fundamental properties of local anesthetics. II. Measured octanol:buffer partition coefficients and pKa values of clinically used drugs

1 reference

12 December 2020

Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin

1 reference

12 December 2020

Specific binding of resiniferatoxin, an ultrapotent capsaicin analog, by dorsal root ganglion membranes

1 reference

12 December 2020

Resiniferatoxin, a phorbol-related diterpene, acts as an ultrapotent analog of capsaicin, the irritant constituent in red pepper

1 reference

12 December 2020

Capsaicin and sensory neurones — a review

1 reference

12 December 2020

The effects of a series of capsaicin analogues on nociception and body temperature in the rat.

1 reference

12 December 2020

Sensory effects of capsaicin congeners. Part II: Importance of chemical structure and pungency in desensitizing activity of capsaicin-type compounds

1 reference

12 December 2020

Effect of capsazepine on the release of calcitonin gene-related peptide-like immunoreactivity (CGRP-LI) induced by low pH, capsaicin and potassium in rat soleus muscle

1 reference

12 December 2020

The role of calcium in capsaicin-induced desensitization in rat cultured dorsal root ganglion neurons

1 reference

12 December 2020

Structure and energetics of ligand binding to proteins: Escherichia coli dihydrofolate reductase-trimethoprim, a drug-receptor system

1 reference

COCI

https://opencitations.net/index/api/v1/references/10.1007/BF00124458

Anti-inflammatory pharmacology and mechanism of the orally active capsaicin analogs, NE-19550 and NE-28345

30 November 2025

1 reference

COCI

https://opencitations.net/index/api/v1/references/10.1007/BF00124458

30 November 2025

Identifiers

DOI

10.1007/BF00124458

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:7561979%20AND%20SRC:MED&resulttype=core&format=json

journals/jcamd/KlopmanL95

20 October 2019

DBLP publication ID

1 reference

DBLP Dataset 2021-01-02

28 January 2021

1 reference