Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin (Q34258414)

31 July 2017

title

Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin (English)

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31 July 2017

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ChEBI release 2020-05-28

1

S. Bevan

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1422598

24 September 2022

author name string

S. Hothi

2

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24 September 2022

G. Hughes

3

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24 September 2022

I. F. James

4

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24 September 2022

H. P. Rang

5

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24 September 2022

K. Shah

6

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24 September 2022

C. S. Walpole

7

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24 September 2022

J. C. Yeats

8

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24 September 2022

publication date

1 October 1992

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https://europepmc.org/articles/PMC1907893

31 July 2017

language of work or name

English

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work available at URL

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1422598

https://europepmc.org/articles/PMC1907893?pdf=render

24 September 2022

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1422598

British Journal of Pharmacology

24 September 2022

published in

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31 July 2017

volume

107

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31 July 2017

issue

2

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31 July 2017

page(s)

544-552

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Sodium and calcium channels in bovine chromaffin cells

31 July 2017

cites work

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Inhibition of human neutrophil 5-lipoxygenase activity by gingerdione, shogaol, capsaicin and related pungent compounds

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Local effector functions of capsaicin-sensitive sensory nerve endings: involvement of tachykinins, calcitonin gene-related peptide and other neuropeptides

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6 July 2018

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Ruthenium red differentiates between capsaicin and nicotine effects on cardiac sensory nerves

6 July 2018

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The antagonism induced by ruthenium red of the actions of capsaicin on the peripheral terminals of sensory neurons: further studies

6 July 2018

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Protective action of ruthenium red toward capsaicin desensitization of sensory fibers

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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Resiniferatoxin, a potent capsaicin-like stimulator of peripheral nociceptors in the neonatal rat tail in vitro

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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Selective antagonism of capsaicin by capsazepine: evidence for a spinal receptor site in capsaicin-induced antinociception

6 July 2018

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6 July 2018

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28 October 2018

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28 October 2018

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28 October 2018

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High affinity insulin binding and insulin receptor-effector coupling: modulation by Ca2+

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12 December 2020

Protons activate a cation conductance in a sub-population of rat dorsal root ganglion neurones

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12 December 2020

Capsaicin causes prolonged inhibition of voltage-activated calcium currents in adult rat dorsal root ganglion neurons in culture

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Inhibitors of calcium buffering depress evoked transmitter release at the squid giant synapse

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A phorbol ester and a daphnane ester stimulate a calcium-independent kinase activity from human mononuclear cells

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Nociceptor stimulation and PGE release by capsaicin

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Antiplatelet effect of capsaicin

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Calcium dependence of baclofen- and GABA-induced depression of responses to transmural stimulation in the guinea-pig isolated ileum

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Effect of ruthenium red on responses mediated by activation of capsaicin-sensitive nerves of the rat urinary bladder

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Antihemostatic and antithrombotic effects of capsaicin in comparison with aspirin and indomethacin

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Calmodulin activation of red blood cell (Ca2+ + Mg2+)-ATPase and its antagonism by phenothiazines

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10.1111/J.1476-5381.1992.TB12781.X

Identifiers

DOI

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31 July 2017

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31 July 2017

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