Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist (Q28379390)

2

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G Valette

3

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G Garcia

4

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L Foulon

5

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G Galindo

6

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L Bankir

7

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B Pouzet

8

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G Guillon

9

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C Barberis

10

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D Chicot

11

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S Jard

12

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P Vilain

13

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C Garcia

14

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E Marty

15

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D Raufaste

16

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G Brossard

17

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D Nisato

18

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J P Maffrand

19

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G Le Fur

Journal of Clinical Investigation

20

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publication date

15 December 1996

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language of work or name

English

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published in

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volume

98

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issue

12

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page(s)

2729-38

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cites work

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Potent aquaretic agent. A novel nonpeptide selective vasopressin 2 antagonist (OPC-31260) in men.

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Syndrome of inappropriate secretion of antidiuretic hormone (SIADH) in malignant disease

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29 September 2017

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Oxytocin release and renal actions in normal and Brattleboro rats

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A radioiodinated linear vasopressin antagonist: a ligand with high affinity and specificity for V1a receptors

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cAMP and extrarenal vasopressin V2 receptors in dogs

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Expression of vasopressin V1a and V2 receptor messenger ribonucleic acid in the liver and kidney of embryonic, developing, and adult rats

2 June 2018

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Vasopressin-induction of cyclic AMP in cultured hippocampal neurons

27 November 2018

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Evidence for the existence of vasopressin V2 receptor mRNA in rat hippocampus

27 November 2018

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Characterization of oxytocin, vasopressin, and neurophysin from the bovine corpus luteum

27 November 2018

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12 December 2020

Stimulation by antidiuretic hormone of electrolyte tubular reabsorption in rat kidney

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12 December 2020

Aquaretic effect of a potent, orally active, nonpeptide V2 antagonist in men

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12 December 2020

Oxytocin as an antidiuretic hormone. II. Role of V2 vasopressin receptor

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12 December 2020

Potent inhibitory effect of SR 49059, an orally active non-peptide vasopressin VIa receptor antagonist, on human arterial coronary bypass graft

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12 December 2020

Autoradiographic localization of vasopressin V1a receptors in the rat kidney using [3H]-SR 49059

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12 December 2020

OPC-21268, an Orally Effective, Nonpeptide Vasopressin V1 Receptor Antagonist

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12 December 2020

Radioligand binding studies reveal marked species differences in the vasopressin V1 receptor of rat, rhesus and human tissues

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12 December 2020

Kinetic and pharmacological characterization of vasopressin membrane receptors from human kidney medulla: Relation to adenylate cyclase activation

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12 December 2020

Vasopressin-, angiotensin II-, and alpha 1-adrenergic-induced inhibition of Ca2+ transport by rat liver plasma membrane vesicles

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12 December 2020